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CDK12-IN-4 [2651196-69-7]

CDK12-IN-4 [2651196-69-7]

T40288
TargetMol Chemicals
CAS Number2651196-69-7
Product group Chemicals
Molecular Weight426.432
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    CDK12-IN-4 [2651196-69-7]
  • Delivery Days Customer
    999
  • CAS Number
    2651196-69-7
  • Category Supplier
    Chemical
  • Certification
    Research Use Only
  • Chemical Name
    CDK12-IN-4
  • Molecular Formula
    C20H20F2N8O
  • Molecular Weight
    426.432
  • Scientific Description
    CDK12-IN-4, a pyrazolotriazine compound, exhibits potent inhibition of CDK12 by achieving an IC50 value of 0.641 microM, utilizing high ATP levels (2 mM). Notably, CDK12-IN-4 does not impact CDK2/Cyclin E (IC50 > 20 microM) or CDK9/Cyclin T1 (IC50 > 20 microM) under the influence of high ATP (2 mM) levels (WO2021116178A1).
  • Shelf life instruction
    3 years
  • SMILES
    Fc1ccc2nc(CNc3nc(nc4c(cnn34)C3CC3)N3CCOCC3)[nH]c2c1F
  • Storage Instruction
    -20°C
  • UNSPSC
    51202000

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