Clobenpropit (dihydrobromide) [145231-35-2]
HY-101198
CAS Number145231-35-2
Product group Chemicals
Estimated Purity99.76
Molecular Weight470.65
Overview
- SupplierMedChem Express
- Product NameClobenpropit (dihydrobromide) [145231-35-2]
- Delivery Days Customer10
- CAS Number145231-35-2
- CertificationResearch Use Only
- Estimated Purity99.76
- Molecular FormulaC14H19Br2ClN4S
- Molecular Weight470.65
- Scientific DescriptionClobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR[1]. Clobenpropit dihydrobromide acts as partial agonist at histamine H4 receptors (Ki 13 nM). Clobenpropit dihydrobromide also binds to serotonin 5-HT3 receptors (Ki 7.4 nM) and alpha2A/alpha2C adrenoceptors (Ki 17.4/7.8 nM)[2]. Clobenpropit dihydrobromide increases apoptosis[3].
- SMILESN=C(SCCCC1=CN=CN1)NCC2=CC=C(Cl)C=C2.[H]Br.[H]Br
- Storage Instruction2°C to 8°C
- UNSPSC12352200
![Clobenpropit dihydrobromide [145231-35-2]](https://www.targetmol.com/group3/M00/02/29/CgoaEGY7KqKEPrtTAAAAAAU7tec016.png)