CP-339818 [185855-91-8]

MedChem Express

CP-339818 [185855-91-8]

9

185855-91-8

Research Use Only

C21H24N2

304.43

CP-339818 is a non-peptide drug with potent Kv1.3 channel blocking activity. CP-339818 is able to effectively inhibit the activation of human T cells. By selectively blocking Kv1.3, CP-339818 is of great value in immune system research. The drug inhibits the C-type inactivated state of Kv1.3 channels in a use-dependent manner. CP-339818 has significantly weaker blocking effects on Kv1.1, Kv1.2, Kv1.5, Kv1.6, Kv3.1-4, and Kv4.2 channels, and only shows some inhibition on the Kv1.4 channel[1].

CCCCC/N=C1C=CN(CC2=CC=CC=C2)C3=C/1C=CC=C3

12352200