Bio-Connect

CPI-0610

ORB1089389
Biorbyt
Molecular Weight365.8129435
Product group Chemicals
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Overview

  • Supplier
    Biorbyt
  • Product Name
    CPI-0610
  • Delivery Days Customer
    10
  • Certification
    Research Use Only
  • Molecular Formula
    C20H16CLN3O2
  • Molecular Weight
    365.8129435
  • Scientific Description
    CPI-0610 is a small molecule inhibitor of the Bromodomain and Extra-Terminal (BET) family of proteins, with potential antineoplastic activity. Upon administration, the BET inhibitor CPI-0610 binds to the acetylated lysine recognition motifs on the bromodomain of BET proteins, thereby preventing the interaction between the BET proteins and acetylated histone peptides. This disrupts chromatin remodeling and gene expression. Prevention of the expression of certain growth-promoting genes may lead to an inhibition of tumor cell growth.
  • SMILES
    ClC1=CC=C(C2=N[C@@]([H])(CC(O)=N)C3ON=C(C)C=3C3=CC=CC=C23)C=C1
  • UNSPSC
    12352200