CPI-169 (racemate)

Biorbyt

CPI-169 (racemate)

16

1450655-76-1

Research Use Only

C27H36N4O5S

528.664

CPI-169 racemate is the racemate form of CPI-169, which is a novel and potent EZH2 inhibitor with IC50 < 1 nM(inhibition of the catalytic activity of PRC2); decreases cellular levels of H3K27me3 with an EC50 of 70 nM, and triggers cell cycle arrest and apo

O=C(C1=C(C)N(C(C2CCN(S(=O)(CC)=O)CC2)C)C3=C1C=CC=C3)NCC4=C(OC)C=C(C)NC4=O

12352200