CPI203 (CPI-203)

Biorbyt

CPI203 (CPI-203) [1446144-04-2]

16

1446144-04-2

Research Use Only

C19H18CLN5OS

399.8971

CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 alpha-screen assay).

ClC1C([H])=C([H])C(=C([H])C=1[H])C1C2C(C([H])([H])[H])=C(C([H])([H])[H])SC=2N2C(C([H])([H])[H])=NN=C2[C@]([H])(C([H])([H])C(N([H])[H])=O)N=1

12352200