CS-2100 [913827-99-3]

MedChem Express

CS-2100 [913827-99-3]

10

913827-99-3

Research Use Only

99.12

C25H23N3O4S

461.53

CS-2100 (Compound 10b) is a potent, selective, orally active and S1P3-sparing S1P1 agonist with an EC50 of 4.0 nM for human S1P1. CS-2100 shows in vivo immunosuppressive efficacy in rats with an ID50 (infective dose) of 0.407 mg/kg for HvGR[1].

O=C(C1CN(CC2=CC(CC)=C(C3=NOC(C4=CC=C(OC5=CC=CC=C5)C=C4)=N3)S2)C1)O

-20°C,2°C to 8°C

12352200