Bio-Connect

CSRM617 (Standard)

HY-122611R
MedChem Express
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Overview

  • Supplier
    MedChem Express
  • Product Name
    CSRM617 (Standard) [787504-88-5]
  • Delivery Days Customer
    5
  • Certification
    Research Use Only
  • Scientific Description
    CSRM617 (Standard) is the analytical standard of CSRM617. This product is intended for research and analytical applications. CSRM617 is a selective small-molecule inhibitor of the transcription factor ONECUT2 (OC2, a master regulator of androgen receptor) with a Kd of 7.43 uM in SPR assays, binding to OC2-HOX domain directly. CSRM617 induces apoptosis by appearance of cleaved Caspase-3 and PARP. CSRM617 is well tolerated in the prostate cancer mouse model [1]
  • UNSPSC
    41116135