CTOP [103429-31-8]

TargetMol Chemicals

CTOP [103429-31-8]

16

103429-31-8

Chemical

Research Use Only

CTOP

C50H67N11O11S2

1062.28

Potent and selective micro opioid receptor antagonist (Ki values are 0.96 and >10,000 nM for micro and delta receptors respectively). Causes behavioral effects on central administration in vivo. Also increases K+ currents in rat locus ceruleus neurons in vitro via a micro receptor independent mechanism.

3 years

C(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=C(O)C=C4)NC(=O)[C@@H](NC([C@@H](CC5=CC=CC=C5)N)=O)CSSC(C)(C)[C@@H](C(N[C@@H]([C@@H](C)O)C(N)=O)=O)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@H](CCCN)NC3=O)[H]

-20°C

12352200