D4R antagonis-2

MedChem Express

D4R antagonis-2 [2846077-70-9]

10

Research Use Only

C21H23ClF2N2O2

408.87

D4R antagonist-2 is a potent and selective D4R antagonist with an IC50 of 6.52 microM. D4R antagonist-2 displays very favorable in vitro PK parameters and has good brain penetration. D4R antagonist-2 has the potential for the research of Parkinsons disease[1].

CC1=C(C=CC=C1NC(CN2CCC(CC2)OCC3=CC=C(C(F)=C3)F)=O)Cl

12131703