Bio-Connect

Deltazinone 1 [894554-89-3]

HY-108436
MedChem Express
CAS Number894554-89-3
Product group Chemicals
Molecular Weight457.57
Sign in to order and to see your custom pricing.
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    MedChem Express
  • Product Name
    Deltazinone 1 [894554-89-3]
  • Delivery Days Customer
    10
  • CAS Number
    894554-89-3
  • Certification
    Research Use Only
  • Molecular Formula
    C27H31N5O2
  • Molecular Weight
    457.57
  • Scientific Description
    Deltazinone 1, a pyrazolopyridazinone, is a highly selective PDEdelta inhibitor with a KD of 8 nM. Deltazinone 1 inhibits the PDEdelta-Ras interaction. Deltazinone 1 shows a dose-dependent inhibitory response on proliferation in oncogenic KRas-dependent cell lines[1][2].
  • SMILES
    CC1=CC=C(N2C(C)=C(C(C)=NN(CCCC(NCC(C)C3=CC=CC=C3)=O)C4=O)C4=N2)C=C1
  • UNSPSC
    12352200