DPM-1001

Biorbyt

DPM-1001 [1471172-27-6]

10

1471172-27-6

Research Use Only

C35H57N3O3

567.8453901

DPM-1001 is a potent, selective, orally bioavailable inhibitor of the protein-tyrosine phosphatase PTP1B with IC50 of 100 nM, also chelates copper, which enhanced its potency as a PTP1B inhibitor.

O[C@@H]1C[C@H]2C[C@@H](CC[C@]2(C)[C@H]2CC[C@]3(C)[C@@H]([C@H](C)CCC(=O)OC)CC[C@H]3[C@@H]21)NCCCCNCC1C=CC=CN=1

12352200