EN4

Biorbyt

EN4 [1197824-15-9]

10

1197824-15-9

Research Use Only

C25H24N2O4

416.4690666

EN4, a covalent ligand that targets cysteine 171 (C171) of MYC, is selective for c-MYC over N-MYC and L-MYC. EN4 inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis.

O(C1C=CC(=CC=1)OCC)C1=CC=CC=C1NC(C1C=CC(=CC=1)CNC(C=C)=O)=O

12352200