Epertinib (hydrochloride)
HY-107367A
CAS Number2071195-74-7
Product group Chemicals
Estimated Purity98.25
Molecular Weight596.48
Overview
- SupplierMedChem Express
- Product NameEpertinib (hydrochloride) [2071195-74-7]
- Delivery Days Customer10
- CAS Number2071195-74-7
- CertificationResearch Use Only
- Estimated Purity98.25
- Molecular FormulaC30H28Cl2FN5O3
- Molecular Weight596.48
- Scientific DescriptionEpertinib (S-22611) hydrochloride is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR , HER4 and HER2 , with IC 50 s of 1.48 nM, 2.49 nM and 7.15 nM, respectively. Epertinib hydrochloride shows potent antitumor activity [1] [2] . Epertinib (hydrochloride) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
- SMILESCC#C/C(C1=CC2=C(NC3=CC=C(OCC4=CC=CC(F)=C4)C(Cl)=C3)N=CN=C2C=C1)=N\OC[C@@H]5NCCOC5.Cl
- Storage Instruction2°C to 8°C
- UNSPSC12352200