EPI-001 [227947-06-0]

HY-100348
Overview
- SupplierMedChem Express
- Product NameEPI-001 [227947-06-0]
- Delivery Days Customer9
- CAS Number227947-06-0
- CertificationResearch Use Only
- Estimated Purity98.87
- Molecular FormulaC21H27ClO5
- Molecular Weight394.89
- Scientific DescriptionEPI-001, a selective inhibitor of Androgen Receptor (AR), targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC50 of ~6 microM. EPI-001 is also a selective modulator of PPARgamma. EPI-001 is active against castration-resistant prostate cancer[1][2][3].
- SMILESOCC(O)COC1=CC=C(C(C)(C2=CC=C(OCC(O)CCl)C=C2)C)C=C1
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200