Bio-Connect

EPI-001 [227947-06-0]

Research Use Only
HY-100348
MedChem Express
CAS Number227947-06-0
Product group Chemicals
Estimated Purity98.87
Molecular Weight394.89
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Overview

  • Supplier
    MedChem Express
  • Product Name
    EPI-001 [227947-06-0]
  • Delivery Days Customer
    9
  • CAS Number
    227947-06-0
  • Certification
    Research Use Only
  • Estimated Purity
    98.87
  • Molecular Formula
    C21H27ClO5
  • Molecular Weight
    394.89
  • Scientific Description
    EPI-001, a selective inhibitor of Androgen Receptor (AR), targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC50 of ~6 microM. EPI-001 is also a selective modulator of PPARgamma. EPI-001 is active against castration-resistant prostate cancer[1][2][3].
  • SMILES
    OCC(O)COC1=CC=C(C(C)(C2=CC=C(OCC(O)CCl)C=C2)C)C=C1
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200