EPZ-719

Biorbyt

EPZ-719 [2697176-16-0]

10

2697176-16-0

Research Use Only

C22H31FN4O3S

450.57

EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0.005 microM) with a high selectivity over other histone methyltransferases.

N1C2=C(C(F)=CC=C2C)C=C1C(N[C@@H]1CCC[C@H](N2CC[C@H](N(C)S(C)(=O)=O)C2)C1)=O

12352200