ERalpha degrader 5

MedChem Express

ERalpha degrader 5 [2941268-96-6]

10

Research Use Only

C29H25F4N3O2S

555.59

ERalpha degrader 5 (Compound 40) is a selective, orally bioavailable estrogen receptor (ER) degrader (SERD) with an EC50 of 1.1 nM against ERalpha. ERalpha degrader 5 shows antitumor effect in vivo[1].

CC(F)(C1=C(C2=C(C3=CC=C4NN=CC4=C3S2)OC5=CC=C(C=C5)OC6CN(C6)CCCF)C=CC(F)=C1)F

12131703