(E/Z)-ZL0420 [2229039-45-4]

MedChem Express

(E/Z)-ZL0420 [2229039-45-4]

10

2229039-45-4

Research Use Only

C16H16N4O2

296.32

(E/Z)-ZL0420 is a racemic compound of (Z)-ZL0420 and (E)-ZL0420 isomers. (E)-ZL0420 is a potent and selective bromodomain-containing protein 4 (BRD4) inhibitor with IC50 values of 27 nM against BRD4 BD1 and 32 nM against BRD4 BD2[1].

O=C1NC2=C(C=C(/N=N/C3=CC(C)=C(O)C=C3N)C=C2)CC1

12352200