Firibastat (Standard) [648927-86-0]
HY-109058R
Product group Assays
Overview
- SupplierMedChem Express
- Product NameFiribastat (Standard) [648927-86-0]
- Delivery Days Customer999
- CertificationResearch Use Only
- Scientific DescriptionFiribastat (Standard) is the analytical standard of Firibastat. This product is intended for research and analytical applications. Firibastat (QGC001), an orally active brain penetrating proagent of EC33, is a first-in-class brain aminopeptidase A (APA) inhibitor (Ki=200 nM). Firibastat selectively and specifically inhibits conversion of brain angiotensin-II into angiotensin-III and decreases blood pressure in hypertensive rats[1][2].
- UNSPSC41116100