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Fonsartan (free acid) [144628-52-4]

HY-119379
MedChem Express
CAS Number144628-52-4
Product group Chemicals
Molecular Weight544.69
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Fonsartan (free acid) [144628-52-4]
  • Delivery Days Customer
    9
  • CAS Number
    144628-52-4
  • Certification
    Research Use Only
  • Molecular Formula
    C26H32N4O5S2
  • Molecular Weight
    544.69
  • Scientific Description
    Fonsartan (HOE-720) free acid is an orally active angiotensin II receptor (AT1R) antagonist with an IC50 value of 0.48 nM, exhibiting potent antihypertensive activity. Fonsartan free acid dose-dependently inhibits angiotensin II-induced pressor response in rats (ID50 = 0.11 mg/kg) and shows significant long-lasting blood pressure-lowering effects in high-renin animal models. Fonsartan free acid is primarily used in research on hypertension and cardiovascular diseases[1].
  • SMILES
    O=C(C1=C(SC)N=C(CCCC)N1CC2=CC=C(C3=C(S(=O)(NC(NCCC)=O)=O)C=CC=C3)C=C2)O
  • UNSPSC
    12352200