Gaboxadol (hydrochloride) (Standard) [85118-33-8]

MedChem Express

Gaboxadol (hydrochloride) (Standard) [85118-33-8]

5

Research Use Only

Gaboxadol (hydrochloride) (Standard) is the analytical standard of Gaboxadol (hydrochloride). This product is intended for research and analytical applications. Gaboxadol hydrochloride (Lu 02-030 hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 microM). Gaboxadol hydrochloride displays a partial agonist efficacy on subunit alpha1beta2gamma2 with an ED50 value of 143 microM, a full agonist efficacy at alpha5 subunit (ED50=28-129 microM) and a superagonist efficacy at alpha4beta3delta (ED50=6 microM). Gaboxadol hydrochloride is a non-opioid agent[1][2].

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