GAT100 [1663564-42-8]

TargetMol Chemicals

GAT100 [1663564-42-8]

86

Research Use Only

GAT100

C25H28N4OS

432.58

GAT100 is a potent and covalent negative allosteric modulator (NAM). GAT-100 behaved as a robust positive allosteric modulator of binding of orthosteric agonist CP55,940. This novel covalent probe can serve as a useful tool for characterizing CB1R allosteric ligand-binding motifs.

3 years

C(C)C=1C=2C(NC1C(NCCC3=CC=C(C=C3)N4CCCCC4)=O)=CC=C(N=C=S)C2

-20°C

12352200