Bio-Connect

GI-530159 [69563-88-8]

HY-W013712
MedChem Express
CAS Number69563-88-8
Product group Chemicals
Estimated Purity99.27
Molecular Weight518.45
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Overview

  • Supplier
    MedChem Express
  • Product Name
    GI-530159 [69563-88-8]
  • Delivery Days Customer
    9
  • CAS Number
    69563-88-8
  • Certification
    Research Use Only
  • Estimated Purity
    99.27
  • Molecular Formula
    C27H20F6N2O2
  • Molecular Weight
    518.45
  • Scientific Description
    GI-530159 is a selective opener of TREK1 and TREK2 potassium channels. GI-530159 displays selectivity for TREK1/2 over TRAAK, TASK3 and other potassium channels, with an EC50 of 0.76 microM for TREK1. GI-530159 reduces rat dorsal root ganglion neuron excitability and shows potential analgesic effect[1].
  • SMILES
    FC(C(C1=CC=C(OC2=CC=C(N)C=C2)C=C1)(C3=CC=C(OC4=CC=C(N)C=C4)C=C3)C(F)(F)F)(F)F
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200