Bio-Connect

Glutaminase-IN-1

HY-114334
MedChem Express
CAS Number2247127-79-1
Product group Chemicals
Estimated Purity98.09
Molecular Weight618.47
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Glutaminase-IN-1 [2247127-79-1]
  • Delivery Days Customer
    10
  • CAS Number
    2247127-79-1
  • Certification
    Research Use Only
  • Estimated Purity
    98.09
  • Molecular Formula
    C26H24F3N7O3Se
  • Molecular Weight
    618.47
  • Scientific Description
    Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA) , with an IC 50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.
  • SMILES
    O=C(NC1=NN=C(CCCCC2=NN=C(NC(CC3=CC=CC(OC(F)(F)F)=C3)=O)C=C2)[Se]1)CC4=NC=CC=C4
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200