Glutaminase-IN-1 [2247127-79-1]

MedChem Express

Glutaminase-IN-1 [2247127-79-1]

10

2247127-79-1

Research Use Only

98.09

C26H24F3N7O3Se

618.47

Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.

O=C(NC1=NN=C(CCCCC2=NN=C(NC(CC3=CC=CC(OC(F)(F)F)=C3)=O)C=C2)[Se]1)CC4=NC=CC=C4

-20°C,2°C to 8°C

12352200