GRPR antagonist-2

MedChem Express

GRPR antagonist-2

10

Research Use Only

C28H32F3N5O4

559.58

GRPR antagonist-2 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 0.77 and 2.5 microM in HGC-27 and Pan02 cells, respectively). Anticancer activity[1].

CC(C)(OC(N1CCN(CC1)C([C@H](CC2=CNC3=C2C=CC=C3)NC(NC4=CC=C(C=C4)C(F)(F)F)=O)=O)=O)C

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