GS-626510 [1637770-13-8]

MedChem Express

GS-626510 [1637770-13-8]

10

1637770-13-8

Research Use Only

99.80

C25H22N4O

394.47

GS-626510 is a potent, and orally active BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively[1].

CC1=C(C2=CC(C3=C4C=CC=NC4=CC=C3C)=C5NC(C6CC6)=NC5=C2)C(C)=NO1

-20°C,2°C to 8°C

12352200