Chemical Structure
GSK-5959
82066
CAS Number901245-65-6
Product group Chemicals
Molecular Weight394.5 Da
Overview
- SupplierBPS Bioscience
- Product NameGSK-5959
- Delivery Days Customer7
- CAS Number901245-65-6
- CertificationResearch Use Only
- Molecular FormulaC22H26N4O3
- Molecular Weight394.5 Da
- Scientific DescriptionGSK-5959 exhibits >100-fold selectivity for BRPF1 (IC50 = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.
- Storage Instruction-20°C
- UNSPSC12352200