GSK-923295

MedChem Express

GSK-923295 [1088965-37-0]

10

1088965-37-0

Research Use Only

99.82

C32H38ClN5O4

592.13

GSK-923295 is a special, allosteric inhibitor of centromere-associated protein-E (CENP-E) kinesin motor ATPase activity, with K i of 3.2+/-0.2 nM and 1.6+/- 0.1 nM for human and canine, respectively.

O=C(N[C@@H](CC1=CC=C(C2=CN3C(C([C@@H](O)C)=CC=C3)=N2)C=C1)CNC(CN(C)C)=O)C4=CC(Cl)=C(C=C4)OC(C)C

-20°C,2°C to 8°C

12352200