GSK1324726A

MedChem Express

GSK1324726A [1300031-52-0]

10

1300031-52-0

Research Use Only

99.75

C25H23ClN2O3

434.91

GSK1324726A is a novel, potent, and selective inhibitor of BET proteins with high affinity to BRD2 ( IC 50 =41 nM), BRD3 ( IC 50 =31 nM), and BRD4 ( IC 50 =22 nM).

ClC1=CC=C(N[C@H]2C3=C(C=CC(C4=CC=C(C(O)=O)C=C4)=C3)N(C(C)=O)[C@@H](C)C2)C=C1

-20°C,2°C to 8°C

12352200