GSK256073 (tris) [1228650-42-7]
HY-119222A
CAS Number1228650-42-7
Product group Chemicals
Molecular Weight377.82
Overview
- SupplierMedChem Express
- Product NameGSK256073 (tris) [1228650-42-7]
- Delivery Days Customer9
- CAS Number1228650-42-7
- CertificationResearch Use Only
- Molecular FormulaC14H24ClN5O5
- Molecular Weight377.82
- Scientific DescriptionGSK256073 tris is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 tris acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia[1][2]. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
- SMILESO=C1NC(N(CCCCC)C2=C1NC(Cl)=N2)=O.OCC(CO)(CO)N
- UNSPSC12352200