GSK2798745

MedChem Express

GSK2798745 [1419609-94-1]

10

1419609-94-1

Research Use Only

99.80

C25H28N6O3

460.53

GSK2798745 is a potent, selective, and orally active transient receptor potential vanilloid 4 ( TRPV4 ) ion channel blocker with IC 50 s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively. GSK2798745 can be used in cardiac and respiratory diseases research [1] [2] [3] .

N#CC1=CC=C2N=CN(C[C@](CCC3)(C)C[C@@]43CN(C5=NC=C(C(C)(O)C)N=C5)C(O4)=O)C2=C1

-20°C,2°C to 8°C

12352200