GSK2801

MedChem Express

GSK2801 [1619994-68-1]

10

1619994-68-1

Research Use Only

99.95

C20H21NO4S

371.45

GSK2801 is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with K d values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4 [1] .

O=C(C)C1=CC(C2=C(S(=O)(C)=O)C=CC=C2)=C3N1C=CC(OCCC)=C3

-20°C,2°C to 8°C

12352200