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GSK3368715 (dihydrochloride)

HY-128717A
MedChem Express
CAS Number1628925-77-8
Product group Chemicals
Estimated Purity99.96
Molecular Weight439.46
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Overview

  • Supplier
    MedChem Express
  • Product Name
    GSK3368715 (dihydrochloride) [1628925-77-8]
  • Delivery Days Customer
    9
  • CAS Number
    1628925-77-8
  • Certification
    Research Use Only
  • Estimated Purity
    99.96
  • Molecular Formula
    C20H40Cl2N4O2
  • Molecular Weight
    439.46
  • Scientific Description
    GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor ( IC 50 =3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) produces a shift in arginine methylation states, alters exon usage, and has strong anti-cancer activity [1] .
  • SMILES
    CNCCN(CC1=CNN=C1C2CCC(COCC)(COCC)CC2)C.Cl.Cl
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200

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