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GSK467

Research Use Only
HY-116761
MedChem Express
CAS Number1628332-52-4
Product group Chemicals
Estimated Purity99.55
Molecular Weight319.32
Price on request
Packing Size
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Overview

  • Supplier
    MedChem Express
  • Product Name
    GSK467 [1628332-52-4]
  • Delivery Days Customer
    10
  • CAS Number
    1628332-52-4
  • Certification
    Research Use Only
  • Estimated Purity
    99.55
  • Molecular Formula
    C17H13N5O2
  • Molecular Weight
    319.32
  • Scientific Description
    GSK467 is a cell penetrant and selective KDM5B (JARID1B or PLU1) inhibitor with a Ki of 10 nM and an IC50 of 26 nM. GSK467 shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members[1][2].
  • SMILES
    O=C1C2=C(NC(OC3=CN(N=C3)CC4=CC=CC=C4)=N1)C=NC=C2
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200