GSK6853

MedChem Express

GSK6853 [1910124-24-1]

10

1910124-24-1

Research Use Only

99.89

C22H27N5O3

409.48

GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. GSK6853 shows excellent BRPF1 potency (pKd=9.5) and greater than 1600-fold selectivity over all other bromodomains[1].

C[C@@H]1CNCCN1C2=C(NC(C3=CC=CC=C3OC)=O)C=C(C(N4C)=C2)N(C)C4=O

-20°C,2°C to 8°C

12352200