Histrelin acetate

Biorbyt

Histrelin acetate [220810-26-4]

16

220810-26-4

C66H86N18O12.NC2H4O2

1383.55

Histrelin is a synthetic gonadotropin-releasing hormone (GNRH) agonist that binds to the GNRH receptor (GNRHR; Ki = 0.2 nM in CHO cells expressing the human receptor).

O=C([C@H](CCC/N=C(/N)\N)NC([C@H](CC(C)C)NC([C@@H](CC1=CN(CC2C=CC=CC=2)C=N1)NC([C@H](CC1C=CC(=CC=1)O)NC([C@H](CO)NC([C@H](CC1=CNC2=CC=CC=C12)NC([C@H](CC1=CN=CN1)NC([C@@H]1CCC(N1)=O)=O)=O)=O)=O)=O)=O)=O)N1CCC[C@H]1C(NCC)=O.OC(C)=O

12352200