I-BET762 carboxylic acid [1300019-38-8]

MedChem Express

I-BET762 carboxylic acid [1300019-38-8]

10

1300019-38-8

Research Use Only

99.55

C20H17ClN4O3

396.83

I-BET762 carboxylic acid (Molibresib carboxylic acid) is an I-BET762-based warhead ligand for conjugation reactions of PROTAC targeting on BET. I-BET762 carboxylic acid (Molibresib carboxylic acid) is a BRD4 inhibitor with a pIC50 of 5.1[1].

CC1=NN=C2[C@H](CC(O)=O)N=C(C3=CC=C(Cl)C=C3)C4=C(C=CC(OC)=C4)N21

-20°C,2°C to 8°C

12352200