J 104129 (fumarate)

MedChem Express

J 104129 (fumarate) [257603-40-0]

5

257603-40-0

Research Use Only

C28H40N2O6

500.63

J 104129 fumarate is a selective and orally active muscarinic M3 antagonist with K i values of 4.2 nM and 490 nM for M3 and M2, respectively. J 104129 fumarate antagonized ACh-induced bronchoconstriction. J 104129 fumarate has the potential for the research of obstructive airway disease [1] .

O=C(NC1CCN(CC/C=C(C)/C)CC1)[C@@](O)(C2CCCC2)C3=CC=CC=C3.OC(/C=C/C(O)=O)=O

12352200