KB SRC 4 [1380088-03-8]

MedChem Express

KB SRC 4 [1380088-03-8]

5

1380088-03-8

Research Use Only

99.22

C32H23ClN8

555.03

KB SRC 4 is a potent, and highly selective c-Src inhibitor, with a Ki of 44 nM and a Kd of 86 nM, and shows no inhibition on c-Abl up to 125 microM; KB SRC 4 has antitumor activity.

NC1=C2C(N(C3=CC=CC(C4=CN=NN4CC5=CC(C6=CC=CC=C6)=CC=C5)=C3)N=C2C7=CC=C(Cl)C=C7)=NC=N1

-20°C,2°C to 8°C

12352200