L-365260 (hemihydrate)

MedChem Express

L-365260 (hemihydrate)

10

Research Use Only

99.75

C24H22N4O2.1/2H2O

407.47

L-365260 hemihydrate is an orally active and selective antagonist of non-peptide gastrin and brain cholecystokinin receptor (CCK-B) , with K i s of 1.9 nM and 2.0 nM, respectively. L-365260 hemihydrate interacts in a stereoselective and competitive manner with guinea pig stomach gastrin and brain CCK receptors [1] [2] [3] .

O=C(NC1=CC=CC(C)=C1)N[C@H]2C(N(C)C3=CC=CC=C3C(C4=CC=CC=C4)=N2)=O.[1/2].O

2°C to 8°C

12352200