L-798106

Biorbyt

L-798106 [244101-02-8]

10

244101-02-8

Research Use Only

C27H22BRNO4S

536.4368854

L-798106 is potent and highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM), it also has micromolar activities at the EP4, EP1 and EP2 receptors with Ki values of 916 nM, > 5000 nM and > 5000 nM at EP4, EP1 and EP2, respectively.

COC1C=CC(Br)=CC=1S(NC(/C=C\C1=CC=CC=C1CC1C=CC2=CC=CC=C2C=1)=O)(=O)=O

12352200