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Lenvatinib

S1164
Selleck Chemicals
CAS Number417716-92-8
Product group Chemicals
Estimated Purity...
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Lenvatinib (E7080) [417716-92-8]
  • Delivery Days Customer
    9
  • CAS Number
    417716-92-8
  • Certification
    Research Use Only
  • Estimated Purity
    ...
  • Scientific Description
    Lenvatinib is a multi-target inhibitor, mostly for VEGFR2(KDR)/VEGFR3(Flt-4) with IC50 of 4 nM/5.2 nM, less potent against VEGFR1/Flt-1, ~10-fold more selective for VEGFR2/3 against FGFR1, PDGFRalpha/beta in cell-free assays. Lenvatinib (E7080) also inhibits FGFR1-4, PDGFR, Kit (c-Kit), RET (c-RET), and shows potent antitumor activities. Phase 3.
  • Storage Instruction
    -80°C
  • UNSPSC
    51202000

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