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LLK203 [2758090-62-7]

HY-162312
MedChem Express
CAS Number2758090-62-7
Product group Chemicals
Estimated Purity98.58
Molecular Weight561.69
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Overview

  • Supplier
    MedChem Express
  • Product Name
    LLK203 [2758090-62-7]
  • Delivery Days Customer
    14
  • CAS Number
    2758090-62-7
  • Certification
    Research Use Only
  • Estimated Purity
    98.58
  • Molecular Formula
    C28H23N3O4S3
  • Molecular Weight
    561.69
  • Scientific Description
    LLK203 is a potent USP2/USP8 dual-target inhibitor with IC50s of 0.89 microM and 0.52 microM, respectively. LLK203 leads a degradation of ERalpha and induces apoptosis of breast cancer MCF-7 cells. LLK203 demonstrates antitumor activities against the 4T1 tumor mice model[1].
  • SMILES
    O=C(C1=CC=C(OC)C=C1NS(=O)(C2=CC=C(C3=CC=C(C)S3)C=C2)=O)NC4=NC(C5=CC=CC=C5)=CS4
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200