Loperamide oxide [106900-12-3]

MedChem Express

Loperamide oxide [106900-12-3]

9

106900-12-3

Research Use Only

C29H33ClN2O3

493.04

Loperamide oxide (R-58425) is a orally active prodrug of the Loperamide (HY-156131). Loperamide oxide incubation with the contents of the intestinal lumen inhibits fluid secretion under aerobic conditions[1][2].

O=C(C(C1=CC=CC=C1)(CC[N@+]2(CC[C@](C3=CC=C(C=C3)Cl)(CC2)O)[O-])C4=CC=CC=C4)N(C)C

12131703