Bio-Connect

LS-104 [368836-72-0]

HY-118084
MedChem Express
CAS Number368836-72-0
Product group Chemicals
Molecular Weight320.34
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Overview

  • Supplier
    MedChem Express
  • Product Name
    LS-104 [368836-72-0]
  • Delivery Days Customer
    9
  • CAS Number
    368836-72-0
  • Certification
    Research Use Only
  • Molecular Formula
    C19H16N2O3
  • Molecular Weight
    320.34
  • Scientific Description
    LS-104 (Tyrene CR-4) is a non-ATP-competitive kinase inhibitor against JAK2, Bcr-Abl and FLT3. LS-104 potently induces apoptosis in JAK2V617F-positive cells and inhibits JAK2 autophosphorylation and downstream signal transduction. LS-104 also inhibits proliferation and induces potent cytotoxic effects in FLT3 expressing leukemic cells. LS-104 is a hydroxystyryl-acrylonitrile compound, which is promising for research of myeloproliferative disorders and refractory/relapsed hematologic malignancies[1][2].
  • SMILES
    OC1=C(O)C=CC(/C=C/C=C(C#N)/C(NCC2=CC=CC=C2)=O)=C1
  • UNSPSC
    12352200