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LT052 [2543545-44-2]

LT052 [2543545-44-2]

T11887
TargetMol Chemicals
CAS Number2543545-44-2
DownloadMSDS
Product group Chemicals
Molecular Weight449.48
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    LT052 [2543545-44-2]
  • Delivery Days Customer
    10
  • CAS Number
    2543545-44-2
  • Category Supplier
    Chemical
  • Certification
    Research Use Only
  • Chemical Name
    LT052
  • Molecular Formula
    C22H19N5O4S
  • Molecular Weight
    449.48
  • Scientific Description
    LT052, a highly active and selective BET BD1 inhibitor with an IC50 of 87.7 nM, demonstrates nanomolar BRD4 BD1 potency and significant selectivity, being 138-fold more selective for BRD4 BD1 over BRD4 BD2 (IC50 =12.130 microM). Its anti-inflammatory properties make it a potential candidate for acute gout arthritis research [1].
  • Shelf life instruction
    3 years
  • SMILES
    COc1ccccc1S(=O)(=O)Nc1ccc2N(C)C(=O)c3cc(nc1c23)-n1cnc(C)c1
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200