Bio-Connect
Mardepodect [898562-94-2]

Mardepodect [898562-94-2]

T16499
TargetMol Chemicals
CAS Number898562-94-2
Product group Chemicals
Estimated Purity99.81%
Molecular Weight392.45
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    Mardepodect [898562-94-2]
  • Delivery Days Customer
    4
  • CAS Number
    898562-94-2
  • Certification
    Research Use Only
  • Chemical Name
    Mardepodect
  • Estimated Purity
    99.81%
  • Molecular Formula
    C25H20N4O
  • Molecular Weight
    392.45
  • Scientific Description
    Mardepodect (PF-2545920) is a phosphodiesterase inhibitor selective for the PDE10A subtype with an IC50 of 0.37 nM and over 1000-fold selectivity over PDE. It is potentially useful for the treatment of schizophrenia. Phosphodiesterase 10A (PDE10A) is highly expressed in striatal medium spiny neurons of both the direct and indirect output pathways. Mardepodect can cross the blood-brain barrier.
  • Shelf life instruction
    3 years
  • SMILES
    Cn1cc(c(n1)-c1ccc(OCc2ccc3ccccc3n2)cc1)-c1ccncc1
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200