Masitinib mesylate

AbMole BioScience

Masitinib mesylate

9

1048007-93-7

Chemical

Research Use Only

C29H34N6O4S2

594.75

Masitinib (AB-1010) mesylate is a potent, orally bioavailable and selective inhibitor of c-Kit, IC50 of 200 nM for human recombinant c-Kit. It also inhibits PDGFRalfa/bèta, LynB with IC50 values of 540, 800 and 510 nM.

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