Bio-Connect

MDR-652 [1933528-96-1]

HY-136363
MedChem Express
CAS Number1933528-96-1
Product group Chemicals
Estimated Purity99.02
Molecular Weight447.95
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Overview

  • Supplier
    MedChem Express
  • Product Name
    MDR-652 [1933528-96-1]
  • Delivery Days Customer
    9
  • CAS Number
    1933528-96-1
  • Certification
    Research Use Only
  • Estimated Purity
    99.02
  • Hazard Information
    h302, h315, h319, h335
  • Molecular Formula
    C22H23ClFN3O2S
  • Molecular Weight
    447.95
  • Scientific Description
    MDR-652 is a highly specific and efficacious transient receptor potential vanilloid 1 (TRPV1) ligand with agonist activity. The Kis are 11.4 and 23.8 nM for hTRPV1 and rTRPV1, respectively. The EC50s are 5.05 and 93 nM for hTRPV1 and rTRPV1, respectively. Potent topical analgesic activity[1].
  • SMILES
    O=C(NC1=CC=C(CO)C(F)=C1)NCC2=C(C3=CC=CC(Cl)=C3)N=C(C(C)(C)C)S2
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200