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Molibresib (I-BET-762) [1260907-17-2]

Research Use Only
S7189
Selleck Chemicals
CAS Number1260907-17-2
Product group Chemicals
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Molibresib (I-BET-762) [1260907-17-2]
  • Delivery Days Customer
    9
  • CAS Number
    1260907-17-2
  • Certification
    Research Use Only
  • Scientific Description
    Molibresib (I-BET-762, GSK525762, GSK525762A) is an inhibitor for BET proteins with IC50 of ~35 nM in a cell-free assay, suppresses the production of proinflammatory proteins by macrophages and blocks acute inflammation, highly selective over other bromodomain-containing proteins.
  • UNSPSC
    12352200

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Chemical Structure
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I-BET-762 [1260907-17-2]
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Molecular Weight423.9 Da
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